Biological Activity
BRD-IN-3 ((R,R)-36n) is a highly potent PCAF bromodomain (BRD) inhibitor, with an IC50 of 7 nM. BRD-IN-3 also exhibits activity against GCN5 and FALZ.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 25.29 mL | 126.44 mL | 252.88 mL |
0.5 mM | 5.06 mL | 25.29 mL | 50.58 mL |
1 mM | 2.53 mL | 12.64 mL | 25.29 mL |
5 mM | 0.51 mL | 2.53 mL | 5.06 mL |
*The above data is based on the productmolecular weight 395.45. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A18454 |
---|---|
Actions | Inhibitor |
M. Wt | 395.45 |
Formula | C21H25N5O3 |
Solubility | DMSO |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 2351938-32-2 |
SMILES | CN(C1)C[[email protected]](NC(N2C)=NC3=C(NC=C3)C2=O)C[[email protected]@H]1C4=CC=C5OCCOC5=C4 |
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