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Brexpiprazole is a novel D2 dopamine partial agonist investigational product currently in clinical trials for the treatment of depression, schizophrenia, and attention deficit hyperactivity disorder (ADHD).
Targets
| 5-HT1A | human noradrenergic α1B | Dopamine D2L | 5-HT2A receptors | α2C receptors |
| 0.12 nM(Ki) | 0.17 nM(Ki) | 0.3 nM(Ki) | 0.47 nM(Ki) | 0.59 nM(Ki) |
| In vitro | DMSO | 21 mg/mL (48.43 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 23.06 mL | 115.32 mL | 230.64 mL |
| 0.5 mM | 4.61 mL | 23.06 mL | 46.13 mL |
| 1 mM | 2.31 mL | 11.53 mL | 23.06 mL |
| 5 mM | 0.46 mL | 2.31 mL | 4.61 mL |
*The above data is based on the productmolecular weight 433.5733. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A13527 |
|---|---|
| Actions | Agonist |
| CAS No. | 913611-97-9 |
| Formula | C25H27N3O2S |
| M. Wt | 433.5733 |
| Purity | >98% |
| Synonyms | OPC 34712, OPC-34712 |
| SMILES | C1CN(CCN1CCCCOC2=CC3=C(C=C2)C=CC(=O)N3)C4=C5C=CSC5=CC=C4 |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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