BX-517

Catalog No.: A12881

PDK1 inhibitor

BX-517

BX-517 Chemical Structure

CAS NO. 850717-64-5

BX-517 is a potent and selective inhibitor of PDK1 that binds to the ATP binding pocket of the protein (IC50 = 6 nM).

Availability: In stock

Package Price Qty
5 mg
$80.00
10 mg
$130.00
25 mg
$290.00
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Biological Activity

BX-517 is a potent and selective inhibitor of PDK1 that binds to the ATP binding pocket of the protein (IC50 = 6 nM).
In vitro DMSO 54 mg/mL (191.29 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 35.42 mL 177.12 mL 354.23 mL
0.5 mM 7.08 mL 35.42 mL 70.85 mL
1 mM 3.54 mL 17.71 mL 35.42 mL
5 mM 0.71 mL 3.54 mL 7.08 mL

*The above data is based on the productmolecular weight 282.3. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12881
Actions Inhibitor
CAS No. 850717-64-5
Formula C15H14N4O2
M. Wt 282.3
Purity >98%
Synonyms BX517, BX 517
SMILES CC(=C1C2=C(C=CC(=C2)NC(=O)N)NC1=O)C3=CC=CN3
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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