Cangrelor Tetrasodium

Catalog No.: A17919

P2Y12 receptors inhibitor

Cangrelor Tetrasodium

Cangrelor Tetrasodium Chemical Structure

CAS NO. 163706-36-3

Cangrelor Tetrasodium is a high-affinity, reversible inhibitor of P2Y12 receptors that causes almost complete inhibition of ADP-induced platelet aggregate. It is a modified ATP derivative stable to enzymatic degradation. Unlike clopidogrel (Plavix), which is a prodrug, cangrelor is an active drug not requiring metabolic conversion.

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5 mg

Regular Price: $350.00

Special Price $280.00

10 mg

Regular Price: $650.00

Special Price $520.00

25 mg

Regular Price: $1,200.00

Special Price $960.00

50 mg

Regular Price: $2,000.00

Special Price $1,600.00

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Biological Activity

Cangrelor Tetrasodium is a high-affinity, reversible inhibitor of P2Y12 receptors that causes almost complete inhibition of ADP-induced platelet aggregate. It is a modified ATP derivative stable to enzymatic degradation. Unlike clopidogrel (Plavix), which is a prodrug, cangrelor is an active drug not requiring metabolic conversion.
In vitro DMSO 2 mg/mL (2.31 mM)
Water 87 mg/mL (100.66 mM)
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 11.57 mL 57.85 mL 115.7 mL
0.5 mM 2.31 mL 11.57 mL 23.14 mL
1 mM 1.16 mL 5.79 mL 11.57 mL
5 mM 0.23 mL 1.16 mL 2.31 mL

*The above data is based on the productmolecular weight 864.27. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A17919
Actions Inhibitor
CAS No. 163706-36-3
Formula C17H21Cl2F3N5Na4O12P3S2
M. Wt 864.27
Solubility DMSO
Purity >98%
Synonyms Cangrelor Tetrasodium; AR-C69931MX; AR C69931MX; ARC69931MX
SMILES CSCCNC1=NC(SCCC(F)(F)F)=NC2=C1N=CN2[[email protected]@H]3O[[email protected]](COP([O-])(OP([O-])(C(P([O-])([O-])=O)(Cl)Cl)=O)=O)[[email protected]@H](O)[[email protected]]3O.[Na+].[Na+].[Na+].[Na+]
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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