Cariprazine

Catalog No.: A21202

D3 receptor and D2 receptor partial agonist

Cariprazine

Cariprazine Chemical Structure

CAS NO. 839712-12-8

Cariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM).

Availability: In stock

Package Price Qty
5 mg
$130.00
10 mg
$223.00
50 mg
$662.00
100 mg
$1,325.00
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Biological Activity

Cariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.4 mL 116.98 mL 233.97 mL
0.5 mM 4.68 mL 23.4 mL 46.79 mL
1 mM 2.34 mL 11.7 mL 23.4 mL
5 mM 0.47 mL 2.34 mL 4.68 mL

*The above data is based on the productmolecular weight 427.41. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21202
Actions Agonist
M. Wt 427.41
Formula C21H32Cl2N4O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 839712-12-8
Synonyms RGH-188, RGH 188, RGH188
SMILES O=C(N[[email protected]]1CC[[email protected]](CCN2CCN(C3=CC=CC(Cl)=C3Cl)CC2)CC1)N(C)C

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