CB1-IN-1

Catalog No.: A59211
Cannabinoid Receptor Antagonist
CB1-IN-1 is a selective cannabinoid receptor type 1 (CB1R) antagonist, demonstrating a potent inhibition with a Ki value of 0. Its peripherally restricted mechanism of action makes it particularly valuable for studies investigating the physiological roles of CB1R in peripheral tissues. CB1-IN-1 is applicable in research focused on metabolic disorders, pain management, and neuroprotection, facilitating the exploration of therapeutic interventions targeting the endocannabinoid system.
Grouped product items
Size Price Stock Qty
1mg
$65.00
In stock
2mg
$95.00
In stock
5mg
$165.00
In stock
10mg
$240.00
In stock
25mg
$395.00
In stock
50mg
$535.00
In stock
100mg
$705.00
In stock
500mg
$1,380.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionCB1-IN-1 is a selective cannabinoid receptor type 1 (CB1R) antagonist, demonstrating a potent inhibition with a Ki value of 0. Its peripherally restricted mechanism of action makes it particularly valuable for studies investigating the physiological roles of CB1R in peripheral tissues. CB1-IN-1 is applicable in research focused on metabolic disorders, pain management, and neuroprotection, facilitating the exploration of therapeutic interventions targeting the endocannabinoid system.
Product Information
Catalog NumA59211
FormulaC33H31Cl2F3N6O3S2
Molecular Weight751.67
CAS Number1429239-98-4
SMILESClC1=CC(Cl)=CC=C1N2C(C3=CC=C(C#CC4=CC=C(C(F)(F)F)C=C4)S3)=C(CNS(=O)(N5CCCC5)=O)C(C(NN6CCCCC6)=O)=N2
SynonymsBPRCB1184
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

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    C2

    V2