CB2R PAM

Catalog No.: A59194
CB2Rs Positive Allosteric Modulator
CB2R PAM is a positive allosteric modulator of cannabinoid type-2 receptors (CB2Rs) with oral bioavailability. This compound exhibits significant antinociceptive activity, demonstrated in vivo in mouse models of neuropathic pain. CB2R PAM offers valuable insights for research applications related to pain management and cannabinoid pharmacology.
Grouped product items
Size Price Stock Qty
1mg
$25.00
In stock
5mg
$60.00
In stock
10mg
$90.00
In stock
25mg
$150.00
In stock
50mg
$220.00
In stock
100mg
$315.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionCB2R PAM is a positive allosteric modulator of cannabinoid type-2 receptors (CB2Rs) with oral bioavailability. This compound exhibits significant antinociceptive activity, demonstrated in vivo in mouse models of neuropathic pain. CB2R PAM offers valuable insights for research applications related to pain management and cannabinoid pharmacology.
Product Information
Catalog NumA59194
FormulaC21H24BrFN2O2
Molecular Weight435.33
CAS Number2244579-87-9
SMILESFC1=CC=C(CN2C(C(NC(C3CCCCCC3)=O)=C(C)C(Br)=C2)=O)C=C1
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