Biological Activity
CCT241533 Hcl is a potent serine/threonine checkpoint kinase (Chk2) inhibitor with IC50 of 3 nM; shows minimal cross-reactivity against a panel of kinases at 1 uM.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 20.88 mL | 104.4 mL | 208.79 mL |
0.5 mM | 4.18 mL | 20.88 mL | 41.76 mL |
1 mM | 2.09 mL | 10.44 mL | 20.88 mL |
5 mM | 0.42 mL | 2.09 mL | 4.18 mL |
*The above data is based on the productmolecular weight 478.94. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A15038 |
---|---|
Actions | Inhibitor |
CAS No. | 1431697-96-9 |
Formula | C23H28ClFN4O4 |
M. Wt | 478.94 |
Purity | >98% |
Synonyms | CCT-241533 hydrochloride, CCT 241533 hydrochloride |
SMILES | CC(C)(C1CNCC1NC2=NC(=C3C=C(C=CC3=O)F)NC4=CC(=C(C=C42)OC)OC)O.Cl |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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