Biological Activity
CCT244747 is a novel potent, highly selective, orally active ATP-competitive CHK1 inhibitor with potential anticancer activity,
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 24.48 mL | 122.41 mL | 244.82 mL |
0.5 mM | 4.9 mL | 24.48 mL | 48.96 mL |
1 mM | 2.45 mL | 12.24 mL | 24.48 mL |
5 mM | 0.49 mL | 2.45 mL | 4.9 mL |
*The above data is based on the productmolecular weight 408.46. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A15550 |
---|---|
Actions | Inhibitor |
M. Wt | 408.46 |
Formula | C20H24N8O2 |
Solubility | DMSO |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 1404095-34-6 |
Synonyms | CCT-244747, CCT 244747 |
SMILES | CC(CN(C)C)OC1=NC(=CN=C1C#N)NC2=NC=C(C(=C2)OC)C3=CN(N=C3)C |
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