CGP 57380

Catalog No.: A13883

MNK2 inhibitor

CGP 57380 Chemical Structure

CAS NO. 522629-08-9

CGP 57380 is an inhibitor of MAP-kinase interacting kinase-1 (Mnk1, MKNK1) (IC50 = 2.2 uM).

Availability: In stock

Package Price Qty
10 mg
$130.00
25 mg
$250.00
50 mg
$400.00
10mM * 1mL in DMSO
$93.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

CGP 57380 is an inhibitor of MAP-kinase interacting kinase-1 (Mnk1, MKNK1) (IC50 = 2.2 uM).
Targets
MNK1
2.2 μM
In vitro DMSO 48 mg/mL heating (196.53 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 40.95 mL 204.73 mL 409.45 mL
0.5 mM 8.19 mL 40.95 mL 81.89 mL
1 mM 4.09 mL 20.47 mL 40.95 mL
5 mM 0.82 mL 4.09 mL 8.19 mL

*The above data is based on the productmolecular weight 244.23. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13883
Actions Inhibitor
M. Wt 244.23
Formula C11H9FN6
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 522629-08-9
Synonyms CGP57380, CGP-57380
SMILES C1=CC(=CC=C1NC2=C3C(=NC=NC3=NN2)N)F

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