CGP36216

Catalog No.: A66873
GABAB Receptor Antagonist
CGP36216 is a selective antagonist of the GABAB receptor, exhibiting a binding affinity with a Ki value of 0.3 μM. This compound is valuable in the study of anxiety and trauma-related disorders, allowing researchers to explore the roles of GABAB receptor modulation in these conditions. Its specificity makes it an important tool for investigating the therapeutic potential of GABAB receptor antagonism in various neuropsychiatric research applications.
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5mg
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50mg
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Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionCGP36216 is a selective antagonist of the GABAB receptor, exhibiting a binding affinity with a Ki value of 0.3 μM. This compound is valuable in the study of anxiety and trauma-related disorders, allowing researchers to explore the roles of GABAB receptor modulation in these conditions. Its specificity makes it an important tool for investigating the therapeutic potential of GABAB receptor antagonism in various neuropsychiatric research applications.
Product Information
Catalog NumA66873
FormulaC5H14NO2P
Molecular Weight151.14
CAS Number123691-29-2
SMILESO=P(CC)(CCCN)O
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