CGP46381

Catalog No.: A66829
GABA Receptor Antagonist
CGP46381 is an orally active GABA receptor antagonist, exhibiting an IC50 of 4.9 μM. It effectively inhibits neuronal depression induced by the application of baclofen. This compound is useful for research applications involving the modulation of GABAB receptor activity and its effects on neuronal signaling.
Grouped product items
Size Price Stock Qty
10mg
$805.00
In stock
50mg
$3,240.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionCGP46381 is an orally active GABA receptor antagonist, exhibiting an IC50 of 4.9 μM. It effectively inhibits neuronal depression induced by the application of baclofen. This compound is useful for research applications involving the modulation of GABAB receptor activity and its effects on neuronal signaling.
Product Information
Catalog NumA66829
FormulaC10H22NO2P
Molecular Weight219.26
CAS Number123691-14-5
SMILESO=P(CC1CCCCC1)(CCCN)O
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