Cipralisant maleate is a selective histamine H3 receptor modulator, exhibiting both antagonistic activity in vivo and agonistic effects in vitro. With a high affinity demonstrated by a pKi of 9.9 and a Ki of 0.47 nM for the rat histamine H3 receptor, this compound shows potential applications in attention-deficit hyperactivity disorder research. Additionally, Cipralisant maleate serves as a click chemistry reagent due to its alkyne group, enabling copper-catalyzed azide-alkyne cycloaddition (CuAAc) with azide-containing molecules.
Cipralisant maleate is a selective histamine H3 receptor modulator, exhibiting both antagonistic activity in vivo and agonistic effects in vitro. With a high affinity demonstrated by a pKi of 9.9 and a Ki of 0.47 nM for the rat histamine H3 receptor, this compound shows potential applications in attention-deficit hyperactivity disorder research. Additionally, Cipralisant maleate serves as a click chemistry reagent due to its alkyne group, enabling copper-catalyzed azide-alkyne cycloaddition (CuAAc) with azide-containing molecules.
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