Clemastine fumarate

Catalog No.: A10226

Histamine Receptor antagonis

Clemastine fumarate

Clemastine fumarate Chemical Structure

CAS NO. 14976-57-9

Clemastine is a selective histamine H1 antagonist. It binds to the histamine H1 receptor, thus blocking the action of endogenous histamine, which leads to temporary relief of the negative symptoms caused by histamine.

Availability: In stock

Package Price Qty
100 mg

Regular Price: $60.00

Special Price $54.00

250 mg

Regular Price: $100.00

Special Price $90.00

10mM * 1mL in DMSO

Regular Price: $62.00

Special Price $55.80

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Clemastine is a selective histamine H1 antagonist. It binds to the histamine H1 receptor, thus blocking the action of endogenous histamine, which leads to temporary relief of the negative symptoms caused by histamine.
Targets
Histamine H1 receptor
3 nM
In vitro (25°C) DMSO 35 mg/mL heating (76.09 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 5 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.74 mL 108.71 mL 217.41 mL
0.5 mM 4.35 mL 21.74 mL 43.48 mL
1 mM 2.17 mL 10.87 mL 21.74 mL
5 mM 0.43 mL 2.17 mL 4.35 mL

*The above data is based on the productmolecular weight 459.96. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10226
Actions N/A
M. Wt 459.96
Formula C21H26ClNO.C4H4O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 14976-57-9
Synonyms meclastin
SMILES C[[email protected]@](C1=CC=CC=C1)(C2=CC=C(C=C2)Cl)OCC[[email protected]]3CCCN3C.C(=C/C(=O)O)\C(=O)O

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