CP-615003 is a potent partial agonist of the GABAA receptor, exhibiting subtype-selectivity with a Ki value of 1.1 μM. This compound is converted into the active metabolite CP-900725 through oxidative deamination, which also shows affinity for the GABAA receptor. Additionally, CP-615003 is a substrate of P-glycoprotein, which may restrict its central nervous system penetration. It is primarily used in research related to CNS disorders and functions of the GABAA receptor.
CP-615003 is a potent partial agonist of the GABAA receptor, exhibiting subtype-selectivity with a Ki value of 1.1 μM. This compound is converted into the active metabolite CP-900725 through oxidative deamination, which also shows affinity for the GABAA receptor. Additionally, CP-615003 is a substrate of P-glycoprotein, which may restrict its central nervous system penetration. It is primarily used in research related to CNS disorders and functions of the GABAA receptor.
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