CP-724714

Catalog No.: A10242

HER2/ErbB2 inhibitor

CP-724714

CP-724714 Chemical Structure

CAS NO. 537705-08-1

CP-724714 is an orally available, small molecule, potent HER-2 tyrosine kinase inhibitor that inhibits HER2 kinase (IC50 3.8 ng/ml) .

Availability: In stock

Package Price Qty
5 mg

Regular Price: $60.00

Special Price $54.00

10 mg

Regular Price: $100.00

Special Price $90.00

25 mg

Regular Price: $230.00

Special Price $207.00

50 mg

Regular Price: $400.00

Special Price $360.00

10mM * 1mL in DMSO

Regular Price: $115.00

Special Price $103.50

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

CP-724714 is an orally available, small molecule, potent HER-2 tyrosine kinase inhibitor that inhibits HER2 kinase (IC50 3.8 ng/ml) .
Targets
HER2/ErbB2 (Cell-free assay)
10 nM
In vitro (25°C) DMSO 94 mg/mL (200.2 mM)
Water <1 mg/mL (<1 mM)
Ethanol 94 mg/mL (200.2 mM)
In vivo 0.5% methylcellulose 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.3 mL 106.5 mL 212.99 mL
0.5 mM 4.26 mL 21.3 mL 42.6 mL
1 mM 2.13 mL 10.65 mL 21.3 mL
5 mM 0.43 mL 2.13 mL 4.26 mL

*The above data is based on the productmolecular weight 469.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10242
Actions Inhibitor
M. Wt 469.5
Formula C27H27N5O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 537705-08-1
Synonyms CP724714
SMILES CC1=NC=C(C=C1)OC2=C(C=C(C=C2)NC3=NC=NC4=C3C=C(C=C4)C=CCNC(=O)COC)C

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