Biological Activity
CPI 0610 is a small molecule inhibitor of the Bromodomain and Extra-Terminal (BET) family of proteins, with potential antineoplastic activity.
Targets
BRD4-BD1 | MYC | |||
39 nM | 180 nM(EC50) |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 27.34 mL | 136.68 mL | 273.36 mL |
0.5 mM | 5.47 mL | 27.34 mL | 54.67 mL |
1 mM | 2.73 mL | 13.67 mL | 27.34 mL |
5 mM | 0.55 mL | 2.73 mL | 5.47 mL |
*The above data is based on the productmolecular weight 365.82. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A16076 |
---|---|
Actions | Inhibitor |
M. Wt | 365.82 |
Formula | C20H16ClN3O2 |
Solubility | DMSO |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 1380087-89-7 |
Synonyms | CPI0610, CPI-0610 |
SMILES | O=C(N)C[[email protected]@H]1N=C(C2=CC=C(Cl)C=C2)C3=CC=CC=C3C4=C1ON=C4C |
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