CPI-169

Catalog No.: A15920

EZH2 inhibitor

CPI-169

CPI-169 Chemical Structure

CAS NO. 1450655-76-1

CPI-169 is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $120.00

Special Price $108.00

10 mg

Regular Price: $180.00

Special Price $162.00

25 mg

Regular Price: $420.00

Special Price $378.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

CPI-169 is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively.
Targets
EZH2 WT EZH2 Y641N EZH1
0.24 nM0.51 nM6.1 nM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.92 mL 94.58 mL 189.16 mL
0.5 mM 3.78 mL 18.92 mL 37.83 mL
1 mM 1.89 mL 9.46 mL 18.92 mL
5 mM 0.38 mL 1.89 mL 3.78 mL

*The above data is based on the productmolecular weight 528.66. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A15920
Actions Inhibitor
M. Wt 528.66
Formula C27H36N4O5S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1450655-76-1
Synonyms CPI 169, CPI169
SMILES CCS(N1CCC([[email protected]@](N2C(C)=C(/C(O)=N/CC(C(O)=N3)=C(OC)C=C3C)C4=CC=CC=C42)([H])C)CC1)(=O)=O

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