CPI-203

Catalog No.: A13068

BET bromodomain Inhibitor

CPI-203

CPI-203 Chemical Structure

CAS NO. 1446144-04-2

CPI203 is a novel potent, selective and cell permeable inhibitor of the bromodomain and extra terminal (BET) family protein BRD4 with an IC50 of ~37 nM (BRD4 α-screen assay).

Availability: In stock

Package Price Qty
5 mg
$90.00
10 mg
$170.00
25 mg
$350.00
50 mg
$550.00
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.
  • Derenzini E, .et al. BET Inhibition-Induced GSK3β Feedback Enhances Lymphoma Vulnerability to PI3K Inhibitors, Cell Rep, 2018, Aug 21;24(8):2155-2166 PMID: 30134175

Biological Activity

CPI203 is a novel potent, selective and cell permeable inhibitor of the bromodomain and extra terminal (BET) family protein BRD4 with an IC50 of ~37 nM (BRD4 α-screen assay).
In vitro DMSO Warmed: 78 mg/mL (195.04 mM)
Water Insoluble
Ethanol 5 mg/mL (12.5 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.01 mL 125.03 mL 250.06 mL
0.5 mM 5 mL 25.01 mL 50.01 mL
1 mM 2.5 mL 12.5 mL 25.01 mL
5 mM 0.5 mL 2.5 mL 5 mL

*The above data is based on the productmolecular weight 399.9. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13068
Actions Inhibitor
CAS No. 1446144-04-2
Formula C19H18ClN5OS
M. Wt 399.9
Purity >98%
Synonyms 0
SMILES CC1=C(SC2=C1C(=N[[email protected]](C3=NN=C(N32)C)CC(=O)N)C4=CC=C(C=C4)Cl)C
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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