CPI-268456

Catalog No.: A15828

CPI-268456

CPI-268456 Chemical Structure

CAS NO. 1380087-86-4

CPI-268456 is a ligand of bromodomain-containing protein 4 (BRD4). It binds to BRD4 (IC50 = <0.5 µM in a cell-free assay) and inhibits LPS-induced IL-6 secretion in THP-1 cells (IC50 = <0.5 µM).

Availability: In stock

Package Price Qty
5 mg
$140.00
10 mg
$250.00
25 mg
$550.00
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Biological Activity

CPI-268456 is a ligand of bromodomain-containing protein 4 (BRD4). It binds to BRD4 (IC50 = <0.5 µM in a cell-free assay) and inhibits LPS-induced IL-6 secretion in THP-1 cells (IC50 = <0.5 µM).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.06 mL 125.3 mL 250.6 mL
0.5 mM 5.01 mL 25.06 mL 50.12 mL
1 mM 2.51 mL 12.53 mL 25.06 mL
5 mM 0.5 mL 2.51 mL 5.01 mL

*The above data is based on the productmolecular weight 399.05. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15828
M. Wt 399.05
Formula C20H15Cl2N3O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1380087-86-4
Synonyms CPI 268456, CPI268456
SMILES C(N)(=O)C[[email protected]@H]1N=C(C2=CC=C(Cl)C=C2)C2=CC(Cl)=CC=C2C2C(C)=NOC=21

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