CPI 4203 is a selective inhibitor of KDM5 demethylases, structurally related to CPI 455 but ~25-fold less potent (IC50 value 250 nM for inhibition of full length KDM5A).
CPI 4203 is a selective inhibitor of KDM5 demethylases, structurally related to CPI 455 but ~25-fold less potent (IC50 value 250 nM for inhibition of full length KDM5A).
Product Information
Catalog Num
A16177
Formula
C16H14N4O
Molecular Weight
278.32
CAS Number
1628214-07-2
SMILES
CCC1=C(N=C2C(=CNN2C1=O)C#N)C3=CC=CC=C3C
Synonyms
CPI-4203, CPI4203
Storage
Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
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