CTEP

Catalog No.: A11968

CTEP

CTEP Chemical Structure

CAS NO. 871362-31-1

CTEP is a highly potent, selective and orally bioavailable allosteric antagonist of mGlu5 receptor with an IC50 of 2.2 nM.

Availability: In stock

Package Price Qty
5 mg
$100.00
10 mg
$180.00
50 mg
$700.00
10mM * 1mL in DMSO
$120.00
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Biological Activity

CTEP is a highly potent, selective and orally bioavailable allosteric antagonist of mGlu5 receptor with an IC50 of 2.2 nM.
Targets
mGlu5
2.2 nM
In vitro (25°C) DMSO 76 mg/mL (193.99 mM)
Water Insoluble
Ethanol 10 mg/mL (25.52 mM)
In vivo 2% DMSO+40% PEG 300+2% Tween 80+ddH2O 8 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.53 mL 127.63 mL 255.25 mL
0.5 mM 5.11 mL 25.53 mL 51.05 mL
1 mM 2.55 mL 12.76 mL 25.53 mL
5 mM 0.51 mL 2.55 mL 5.11 mL

*The above data is based on the productmolecular weight 391.77. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11968
CAS No. 871362-31-1
Formula C19H13ClF3N3O
M. Wt 391.77
Purity >98%
SMILES CC1=C(N=C(N1C2=CC=C(C=C2)OC(F)(F)F)C)C#CC3=CC(=NC=C3)Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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