Cyprodime

Catalog No.: A62395
MOR Antagonist
Cyprodime is a selective μ opioid receptor (MOR) antagonist with a Ki value of 5.4 nM for MOR, and significantly lower affinities for δ and κ receptors, measuring 244.6 nM and 2187 nM, respectively. This compound is primarily utilized in research to investigate the role of MOR in pain modulation, addiction studies, and the exploration of opioid receptor pathways. Cyprodime serves as a valuable tool in pharmacological studies aimed at understanding the nuances of opioid receptor signaling.
Grouped product items
Size Price Stock Qty
5mg
$350.00
In stock
10mg
$650.00
In stock
50mg
$2,000.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
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Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
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Biological Activity
DescriptionCyprodime is a selective μ opioid receptor (MOR) antagonist with a Ki value of 5.4 nM for MOR, and significantly lower affinities for δ and κ receptors, measuring 244.6 nM and 2187 nM, respectively. This compound is primarily utilized in research to investigate the role of MOR in pain modulation, addiction studies, and the exploration of opioid receptor pathways. Cyprodime serves as a valuable tool in pharmacological studies aimed at understanding the nuances of opioid receptor signaling.
Product Information
Catalog NumA62395
FormulaC22H29NO3
Molecular Weight355.47
CAS Number118111-54-9
SMILESCO[C@@]12[C@]3(CC(CC2)=O)C4=C(OC)C=CC=C4C[C@@]1([H])N(CC5CC5)CC3
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