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Darapladib analog-1

Catalog No.: A77216
Darapladib Analog
Darapladib analog-1 is an O-alkylated derivative of Darapladib that specifically targets lipoprotein-associated phospholipase A2 (Lp-PLA2). This compound exhibits potent inhibitory activity against Lp-PLA2, making it a valuable reagent for studying the pathophysiology of atherosclerosis. Researchers can utilize Darapladib analog-1 to explore its therapeutic potential in cardiovascular disease development and progression.
Darapladib analog-1 1389264-17-8 Darapladib Analog
Grouped product items
Size Price Stock Qty
1mg
$95.00
In stock
5mg
$220.00
In stock
10mg
$330.00
In stock
25mg
$495.00
In stock
50mg
$680.00
In stock
100mg
$905.00
In stock
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Research use only. We do not sell to patients.
Data Sheet SDS

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionDarapladib analog-1 is an O-alkylated derivative of Darapladib that specifically targets lipoprotein-associated phospholipase A2 (Lp-PLA2). This compound exhibits potent inhibitory activity against Lp-PLA2, making it a valuable reagent for studying the pathophysiology of atherosclerosis. Researchers can utilize Darapladib analog-1 to explore its therapeutic potential in cardiovascular disease development and progression.
Product Information
Catalog NumA77216
FormulaC36H38F4N4O2S
Molecular Weight666.77
CAS Number1389264-17-8
SMILESO=C(COC1=NC(SCC2=CC=C(C=C2)F)=NC3=C1CCC3)N(CCN(CC)CC)CC4=CC=C(C5=CC=C(C(F)(F)F)C=C5)C=C4
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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Metabolism > Phospholipases