Darbufelone mesylate

Name: Darbufelone mesylate
Brand: Adooq Bioscience
SKU: A11789
Rating: 5 (288 reviews)

Catalog No.: A11789

PGF2α/LTB4 production inhibitor

Darbufelone mesylate (CI-1004 mesylate) is a dual inhibitor of cellular PGF2α and LTB4 production. Darbufelone potently inhibits PGHS-2 (IC50 = 0.19 μM) but is much less potent with PGHS-1 (IC50= 20 μM).

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Darbufelone mesylate 139340-56-0 PGF2α/LTB4 production inhibitor

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Grouped product items
Size	Price	Stock
1mg	$55.00	In stock
5mg	$115.00	In stock
10mg	$215.00	In stock
25mg	$450.00	In stock
50mg	$775.00	In stock
100mg	$1,315.00	In stock
Bulk Size	Bulk Discount

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Data Sheet SDS

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Biological Activity

Description	Darbufelone mesylate (CI-1004 mesylate) is a dual inhibitor of cellular PGF2α and LTB4 production. Darbufelone potently inhibits PGHS-2 (IC50 = 0.19 μM) but is much less potent with PGHS-1 (IC50= 20 μM).

Product Information

Catalog Num	A11789
Formula	C19H28N2O5S2
Molecular Weight	428.57
CAS Number	139340-56-0
SMILES	O=C1N=C(N)S/C1=C\C2=CC(C(C)(C)C)=C(O)C(C(C)(C)C)=C2.CS(=O)(O)=O
Synonyms	CI-1004 mesylate
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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