DG172 dihydrochloride

Catalog No.: A16309

PPARβ/δ inverse agonist

DG172 dihydrochloride

DG172 dihydrochloride Chemical Structure

CAS NO. 1361504-77-9

DG-172 is an orally active potent PPARβ/δ inverse agonist (IC50 = 26.9 nM). DG-172 inhibits Angptl4 gene expression in mouse myoblasts (IC50 = 9.5 nM) in vitro.

Availability: In stock

Package Price Qty
5 mg
$50.00
10 mg
$90.00
50 mg
$360.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

DG-172 is an orally active potent PPARβ/δ inverse agonist (IC50 = 26.9 nM). DG-172 inhibits Angptl4 gene expression in mouse myoblasts (IC50 = 9.5 nM) in vitro.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.97 mL 109.84 mL 219.67 mL
0.5 mM 4.39 mL 21.97 mL 43.93 mL
1 mM 2.2 mL 10.98 mL 21.97 mL
5 mM 0.44 mL 2.2 mL 4.39 mL

*The above data is based on the productmolecular weight 455.22. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A16309
Actions Antagonist
M. Wt 455.22
Formula C20H22BrCl2N3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1361504-77-9
Synonyms DG 172 dihydrochloride
SMILES N#C/C(C1=CC=CC=C1Br)=C\C2=CC=C(N3CCN(C)CC3)C=C2.[H]Cl.[H]Cl

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