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Diazepinomicin, also known as TLN-4601, is a small-molecule inhibitor of the RAS/RAF/MAPK signaling pathway with potential antineoplastic activity.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 21.62 mL | 108.09 mL | 216.18 mL |
| 0.5 mM | 4.32 mL | 21.62 mL | 43.24 mL |
| 1 mM | 2.16 mL | 10.81 mL | 21.62 mL |
| 5 mM | 0.43 mL | 2.16 mL | 4.32 mL |
*The above data is based on the productmolecular weight 462.58. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A12891 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 733035-26-2 |
| Formula | C28H34N2O4 |
| M. Wt | 462.58 |
| Purity | >98% |
| Synonyms | TLN-4601; ECO 4601; BU 4664L; ECO 04601 |
| SMILES | CC(=CCC/C(=C/CC/C(=C/CN1C2=CC(=CC(=C2NC3=C(C1=O)C=CC=C3O)O)O)/C)/C)C |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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