EI1

Catalog No.: A12711

EZH2 inhibitor

EI1

EI1 Chemical Structure

CAS NO. 1418308-27-6

EI1 is a potent and selective small molecule inhibitor of EZH2 with IC50 values of 15 nM and 13 nM for wild type EZH2 and EZH2 Y641F mutant, respectively.

Availability: In stock

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5 mg

Regular Price: $95.00

Special Price $76.00

10 mg

Regular Price: $160.00

Special Price $128.00

50 mg

Regular Price: $480.00

Special Price $384.00

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Biological Activity

EI1 is a potent and selective small molecule inhibitor of EZH2 with IC50 values of 15 nM and 13 nM for wild type EZH2 and EZH2 Y641F mutant, respectively.
In vitro DMSO Warmed: 39 mg/mL (99.87 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.61 mL 128.05 mL 256.1 mL
0.5 mM 5.12 mL 25.61 mL 51.22 mL
1 mM 2.56 mL 12.8 mL 25.61 mL
5 mM 0.51 mL 2.56 mL 5.12 mL

*The above data is based on the productmolecular weight 390.48. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12711
Actions Inhibitor
CAS No. 1418308-27-6
Formula C23H26N4O2
M. Wt 390.48
Purity >98%
Synonyms Ezh2 inhibitor, EI-1, EI 1
SMILES CCC(CC)N1C=CC2=C(C=C(C=C21)C#N)C(=O)NCC3=C(C=C(NC3=O)C)C
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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