Enasidenib

Catalog No.: A15808

IDH2 inhibitor

Enasidenib

Enasidenib Chemical Structure

CAS NO. 1446502-11-9

Enasidenib is a potent and selective IDH2 inhibitor with potential anticancer activity (IDH2 = Isocitrate dehydrogenase 2).

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5 mg

Regular Price: $75.00

Special Price $60.00

10 mg

Regular Price: $120.00

Special Price $96.00

25 mg

Regular Price: $210.00

Special Price $168.00

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Biological Activity

Enasidenib is a potent and selective IDH2 inhibitor with potential anticancer activity (IDH2 = Isocitrate dehydrogenase 2).
Targets
IDH2
12 nM
In vitro DMSO 90 mg/mL (190.12 mM)
Water Insoluble
Ethanol 90 mg/mL (190.12 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.12 mL 105.62 mL 211.25 mL
0.5 mM 4.22 mL 21.12 mL 42.25 mL
1 mM 2.11 mL 10.56 mL 21.12 mL
5 mM 0.42 mL 2.11 mL 4.22 mL

*The above data is based on the productmolecular weight 473.38. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15808
Actions Inhibitor
CAS No. 1446502-11-9
Formula C19H17F6N7O
M. Wt 473.38
Purity >98%
Synonyms AG-221, AG 221, AG221
SMILES CC(C)(CNC1=NC(=NC(=N1)NC2=CC(=NC=C2)C(F)(F)F)C3=NC(=CC=C3)C(F)(F)F)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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