EPI-001

Catalog No.: A15814
Androgen Receptor antagonist
EPI-001 is an antagonist of the androgen receptor (AR) that acts by binding covalently to the N-terminal domain (NTD) of the AR and blocking protein-protein interactions required for transcriptional activity of the AR and its splice variants (IC50 for inhibition of AR NTD transactivation ?? 6 μM)
Grouped product items
Product Name Price Stock Qty
EPI-001 10mg
$70.00
In stock
EPI-001 25mg
$150.00
In stock
EPI-001 50mg
$210.00
In stock
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Biological Activity
Discription EPI-001 is an antagonist of the androgen receptor (AR) that acts by binding covalently to the N-terminal domain (NTD) of the AR and blocking protein-protein interactions required for transcriptional activity of the AR and its splice variants (IC50 for inhibition of AR NTD transactivation ?? 6 μM)
Targets
Target Value
Product Information
Catalog Num A15814
Formula C21H27ClO5
Molecular Weight 394.89
CAS Number 227947-06-0
SMILES CC(C)(C1=CC=C(C=C1)OCC(CO)O)C2=CC=C(C=C2)OCC(CCl)O
Synonyms EPI001, EPI 001
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro DMSO 72 mg/mL (182.32 mM)
Water Insoluble
Ethanol 72 mg/mL (182.32 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.32 mL 126.62 mL 253.24 mL
0.5 mM 5.06 mL 25.32 mL 50.65 mL
1 mM 2.53 mL 12.66 mL 25.32 mL
5 mM 0.51 mL 2.53 mL 5.06 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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