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Biological Activity
EPI-001 is an antagonist of the androgen receptor (AR) that acts by binding covalently to the N-terminal domain (NTD) of the AR and blocking protein-protein interactions required for transcriptional activity of the AR and its splice variants (IC50 for inhibition of AR NTD transactivation ?? 6 μM)
Targets
| PPARγ | Androgen Receptor | |||
| N/A | 6 μM |
| In vitro | DMSO | 72 mg/mL (182.32 mM) | |
| Water | Insoluble | ||
| Ethanol | 72 mg/mL (182.32 mM) | ||
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 25.32 mL | 126.62 mL | 253.24 mL |
| 0.5 mM | 5.06 mL | 25.32 mL | 50.65 mL |
| 1 mM | 2.53 mL | 12.66 mL | 25.32 mL |
| 5 mM | 0.51 mL | 2.53 mL | 5.06 mL |
*The above data is based on the productmolecular weight 394.89. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A15814 |
|---|---|
| Actions | Antagonist |
| CAS No. | 227947-06-0 |
| Formula | C21H27ClO5 |
| M. Wt | 394.89 |
| Purity | >98% |
| Synonyms | EPI001, EPI 001 |
| SMILES | CC(C)(C1=CC=C(C=C1)OCC(CO)O)C2=CC=C(C=C2)OCC(CCl)O |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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