EPI-001

Catalog No.: A15814

Androgen Receptor antagonist

EPI-001

EPI-001 Chemical Structure

CAS NO. 227947-06-0

EPI-001 is an antagonist of the androgen receptor (AR) that acts by binding covalently to the N-terminal domain (NTD) of the AR and blocking protein-protein interactions required for transcriptional activity of the AR and its splice variants (IC50 for inhibition of AR NTD transactivation ?? 6 μM)

Availability: In stock

Package Price Qty
10 mg

Regular Price: $70.00

Special Price $56.00

25 mg

Regular Price: $150.00

Special Price $120.00

50 mg

Regular Price: $210.00

Special Price $168.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Details

EPI-001 is an antagonist of the androgen receptor (AR) that acts by binding covalently to the N-terminal domain (NTD) of the AR and blocking protein-protein interactions required for transcriptional activity of the AR and its splice variants (IC50 for inhibition of AR NTD transactivation ?? 6 μM)
Targets
PPARγ Androgen Receptor
N/A6 μM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.32 mL 126.62 mL 253.24 mL
0.5 mM 5.06 mL 25.32 mL 50.65 mL
1 mM 2.53 mL 12.66 mL 25.32 mL
5 mM 0.51 mL 2.53 mL 5.06 mL

*The above data is based on the productmolecular weight 394.89. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

Catalog Num A15814
Actions Antagonist
M. Wt 394.89
Formula C21H27ClO5
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 227947-06-0
Synonyms EPI001, EPI 001
SMILES CC(C)(C1=CC=C(C=C1)OCC(CO)O)C2=CC=C(C=C2)OCC(CCl)O

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