EPZ-5676 (Pinometostat)

Catalog No.: A12735

DOT1L Inhibitor‎

EPZ-5676 (Pinometostat)

EPZ-5676 (Pinometostat) Chemical Structure

CAS NO. 1380288-87-8

EPZ-5676 is a small molecule inhibitor of histone methyltransferase with potential antineoplastic activity.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $80.00

Special Price $64.00

10 mg

Regular Price: $150.00

Special Price $120.00

25 mg

Regular Price: $300.00

Special Price $240.00

50 mg

Regular Price: $500.00

Special Price $400.00

10mM * 1mL in DMSO
$149.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Details

EPZ-5676 is a small molecule inhibitor of histone methyltransferase with potential antineoplastic activity.
Targets
DOT1L (Cell-free assay)
80 pM(Ki)
In vitro (25°C) DMSO 100 mg/mL (177.71 mM)
Water <1 mg/mL (<1 mM)
Ethanol 100 mg/mL (177.71 mM)
In vivo 30% PEG400/0.5% Tween80/5% propylene glycol 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.77 mL 88.86 mL 177.71 mL
0.5 mM 3.55 mL 17.77 mL 35.54 mL
1 mM 1.78 mL 8.89 mL 17.77 mL
5 mM 0.36 mL 1.78 mL 3.55 mL

*The above data is based on the productmolecular weight 562.7. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

Catalog Num A12735
Actions Inhibitor
M. Wt 562.7
Formula C30H42N8O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1380288-87-8
Synonyms EPZ5676, EPZ 5676
SMILES CC(C)N(C[[email protected]@H]1[[email protected]]([[email protected]]([[email protected]@H](O1)N2C=NC3=C2N=CN=C3N)O)O)C4CC(C4)CCC5=NC6=C(N5)C=C(C=C6)C(C)(C)C

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