EPZ020411 hydrochloride

Catalog No.: A21802

PRMT6 inhibitor

EPZ020411 hydrochloride

EPZ020411 hydrochloride Chemical Structure

CAS NO. 2070015-25-5

EPZ020411 hydrochloride is a potent and selective inhibitor of PRMT6 with IC50 of 10 nM, has ??10 fold selectivity for PRMT6 over PRMT1 and PRMT8.

Availability: In stock

Package Price Qty
5 mg
$135.00
10 mg
$233.00
50 mg
$690.00
100 mg
$1,380.00
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Biological Activity

EPZ020411 hydrochloride is a potent and selective inhibitor of PRMT6 with IC50 of 10 nM, has ??10 fold selectivity for PRMT6 over PRMT1 and PRMT8.
In vitro DMSO 86 mg/mL (166.81 mM)
Water 70 mg/mL (135.78 mM)
Ethanol 86 mg/mL (166.81 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.87 mL 104.37 mL 208.74 mL
0.5 mM 4.17 mL 20.87 mL 41.75 mL
1 mM 2.09 mL 10.44 mL 20.87 mL
5 mM 0.42 mL 2.09 mL 4.17 mL

*The above data is based on the productmolecular weight 479.06. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21802
Actions Inhibitor
CAS No. 2070015-25-5
Formula C25H39ClN4O3
M. Wt 479.06
Purity >98%
Synonyms EPZ-020411, EPZ 020411
SMILES CNCCN(C)CC1=CNN=C1C2=CC=C(O[[email protected]]3C[[email protected]](OCCC4CCOCC4)C3)C=C2.Cl[H]
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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