ERG-IN-5

Name: ERG-IN-5
Brand: Adooq Bioscience
SKU: A68263
Rating: 5 (288 reviews)

Catalog No.: A68263

hERG Inhibitor

ERG-IN-5 is a potent hERG potassium channel inhibitor, demonstrating an IC50 value of 1.5 μM. This compound exhibits significant cytotoxicity towards MTAPdel HCT116 cells, with a CC50 of 28 nM. ERG-IN-5 is valuable for research applications focused on colon cancer, facilitating the exploration of mechanisms related to potassium channel modulation and cancer cell viability.

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Biological Activity

Description	ERG-IN-5 is a potent hERG potassium channel inhibitor, demonstrating an IC50 value of 1.5 μM. This compound exhibits significant cytotoxicity towards MTAPdel HCT116 cells, with a CC50 of 28 nM. ERG-IN-5 is valuable for research applications focused on colon cancer, facilitating the exploration of mechanisms related to potassium channel modulation and cancer cell viability.

Product Information

Catalog Num	A68263
Formula	C23H20F3N7O2
Molecular Weight	483.45
CAS Number	3047675-62-4
SMILES	NC1=NC(C=CC(C(N(NC(C2CC2)=O)CC3=NC=C(C(F)(F)F)C=C3)=O)=C4)=C4C5=C1C=NN5C

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