ERRγ inverse agonist 1

Catalog No.: A85305
Estrogen Receptor/ERR Antagonist
ERRγ Inverse Agonist 1 is a selective inverse agonist of the estrogen-related receptor gamma (ERRγ) with an IC50 value of 40 nM. This compound exhibits potent antagonistic activity, making it useful for investigating the role of ERRγ in various biological processes. It is particularly relevant for research applications focused on metabolic regulation and cancer biology, where modulation of ERRγ signaling is of interest.
Grouped product items
Size Price Stock Qty
25mg
$1,275.00
In stock
50mg
$1,625.00
In stock
100mg
$2,000.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

Loading distributor info...

Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionERRγ Inverse Agonist 1 is a selective inverse agonist of the estrogen-related receptor gamma (ERRγ) with an IC50 value of 40 nM. This compound exhibits potent antagonistic activity, making it useful for investigating the role of ERRγ in various biological processes. It is particularly relevant for research applications focused on metabolic regulation and cancer biology, where modulation of ERRγ signaling is of interest.
Product Information
Catalog NumA85305
FormulaC30H38Cl2N2O2
Molecular Weight529.54
CAS Number2316832-86-5
SMILESOC1=CC=CC(/C(C2=CC=C(N3CCN(C(C)C)CC3)C=C2)=C(C4=CC=CC=C4)\CCCO)=C1.[H]Cl.[H]Cl
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

  • Mass

    Concentration

    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

    V1

    C2

    V2