EST73502 is a selective dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, demonstrating effective blood-brain barrier penetration. With binding affinities (Kis) of 64 nM for MOR and 118 nM for σ1R, EST73502 exhibits notable antinociceptive properties. This compound is pertinent for research applications in pain management and neurological studies, allowing for the exploration of opioid receptor pathways and σ1R interactions.
EST73502 is a selective dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, demonstrating effective blood-brain barrier penetration. With binding affinities (Kis) of 64 nM for MOR and 118 nM for σ1R, EST73502 exhibits notable antinociceptive properties. This compound is pertinent for research applications in pain management and neurological studies, allowing for the exploration of opioid receptor pathways and σ1R interactions.
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