Glimepiride

Catalog No.: A10430

Kir6.2/SUR inhibitor

Glimepiride

Glimepiride Chemical Structure

CAS NO. 93479-97-1

Glimepiride is a potent Kir6.2/SUR inhibitor with IC50 of 3.0 nM, 5.4 nM, and 7.3 nM for SUR1, SUR2A and SUR2B, used in the treatment of type 2 diabetes mellitus.

Availability: In stock

Package Price Qty
500 mg
$60.00
1000 mg
$100.00
2000 mg
$180.00
5000 mg
$400.00
10mM * 1mL in DMSO
$60.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Glimepiride is a potent Kir6.2/SUR inhibitor with IC50 of 3.0 nM, 5.4 nM, and 7.3 nM for SUR1, SUR2A and SUR2B, used in the treatment of type 2 diabetes mellitus.
Targets
SUR1 SUR2A SUR2B
3 nM5.4 nM7.3 nM
In vitro DMSO 11 mg/mL (22.42 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.38 mL 101.91 mL 203.82 mL
0.5 mM 4.08 mL 20.38 mL 40.76 mL
1 mM 2.04 mL 10.19 mL 20.38 mL
5 mM 0.41 mL 2.04 mL 4.08 mL

*The above data is based on the productmolecular weight 490.62. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10430
Actions Inhibitor
M. Wt 490.62
Formula C24H34N4O5S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 93479-97-1
Synonyms Amary
SMILES CCC1=C(CN(C1=O)C(=O)NCCC2=CC=C(C=C2)S(=O)(=O)NC(=O)NC3CCC(CC3)C)C

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy Glimepiride | Glimepiride Supplier | purchase | cost | manufacturer | order | distributor | buy 93479-97-1| 93479-97-1 Supplier | purchase 93479-97-1 | 93479-97-1 cost | 93479-97-1 manufacturer | order 93479-97-1 | 93479-97-1 distributor
Rewards