GNA002

Catalog No.: A13266

covalent EZH2 inhibitor

GNA002

GNA002 Chemical Structure

CAS NO. 1385035-79-9

GNA002 is a highly potent, specific and covalent EZH2 (Enhancer of zeste homolog 2) inhibitor with an IC50 of 1.1 μM.

Availability: In stock

Package Price Qty
1 mg
$320.00
5 mg
$960.00
10 mg
$1,600.00
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Biological Activity

GNA002 is a highly potent, specific and covalent EZH2 (Enhancer of zeste homolog 2) inhibitor with an IC50 of 1.1 μM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 14.25 mL 71.24 mL 142.47 mL
0.5 mM 2.85 mL 14.25 mL 28.49 mL
1 mM 1.42 mL 7.12 mL 14.25 mL
5 mM 0.28 mL 1.42 mL 2.85 mL

*The above data is based on the productmolecular weight 701.89. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13266
Actions Inhibitor
M. Wt 701.89
Formula C42H55NO8
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1385035-79-9
Synonyms GNA 002, GNA-002
SMILES O=C(NCCOCC)/C(C)=C\C[[email protected]@]1(C2=O)OC(C)(C)[[email protected]]([[email protected]]31OC4=C5C(O)=C(C/C=C(C)/CC/C=C(C)\C)C(O)=C4C/C=C(C)\C)([H])C[[email protected]@]2([H])C=C3C5=O

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