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Biological Activity
GNE-616 is a highly potent, metabolically stable, orally bioavailable, and subtype selective Nav1.7 inhibitor (Ki of 0.79 nM and Kd of 0.38 nM for hNav1.7) for the treatment of chronic pain.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 18.6 mL | 93.02 mL | 186.04 mL |
| 0.5 mM | 3.72 mL | 18.6 mL | 37.21 mL |
| 1 mM | 1.86 mL | 9.3 mL | 18.6 mL |
| 5 mM | 0.37 mL | 1.86 mL | 3.72 mL |
*The above data is based on the productmolecular weight 537.53. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A19046 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 2349371-81-7 |
| Formula | C24H23F4N5O3S |
| M. Wt | 537.53 |
| Purity | >98% |
| Synonyms | GNE 616, GNE616 |
| SMILES | O=S(C1=C(F)C=C2[[email protected]@H](N3[[email protected]@H](C4=NC=CC=C4)C[[email protected]@H](C(F)(F)F)CC3)CCOC2=C1)(NC5=NC=NC=C5)=O |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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