GPER activator 1

Catalog No.: A85190
GPER activator
GPER Activator 1 is a selective activator of the G protein-coupled estrogen receptor (GPER). This compound has been shown to exhibit dual inhibition of inflammation induced by TNFα and IL-6, making it a valuable tool for investigating the role of GPER in inflammatory responses. Its non-cytotoxic nature further supports its application in various biological research settings.
Grouped product items
Size Price Stock Qty
25mg
$1,655.00
In stock
50mg
$2,115.00
In stock
100mg
$2,720.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionGPER Activator 1 is a selective activator of the G protein-coupled estrogen receptor (GPER). This compound has been shown to exhibit dual inhibition of inflammation induced by TNFα and IL-6, making it a valuable tool for investigating the role of GPER in inflammatory responses. Its non-cytotoxic nature further supports its application in various biological research settings.
Product Information
Catalog NumA85190
FormulaC17H14ClFN2O2S
Molecular Weight364.82
CAS Number2629960-35-4
SMILESCC1=C(C(C)=C(C(NC(C2=C(C3=C(S2)C=C(F)C=C3)Cl)=O)=N1)C)O
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