GR-175737

Catalog No.: A34170
Partial Histamine H3 Receptor Agonist
GR-175737 is a partial agonist of the histamine H3 receptor, exhibiting an EC50 value of 7.8 nM. This compound is primarily utilized in research focused on inflammatory diseases, facilitating the investigation of H3 receptor modulation in various pathophysiological contexts. Its pharmacological profile makes it a valuable tool for studying the role of histamine receptors in inflammation and related disorders.
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Size Price Stock Qty
25mg
$1,275.00
In stock
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Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionGR-175737 is a partial agonist of the histamine H3 receptor, exhibiting an EC50 value of 7.8 nM. This compound is primarily utilized in research focused on inflammatory diseases, facilitating the investigation of H3 receptor modulation in various pathophysiological contexts. Its pharmacological profile makes it a valuable tool for studying the role of histamine receptors in inflammation and related disorders.
Product Information
Catalog NumA34170
FormulaC14H13ClN4O
Molecular Weight288.73
CAS Number176860-26-7
SMILESClC1=CC=C(C=C1)CC2=NOC(CCC3=CN=CN3)=N2
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