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GSK 1210151A (I-BET151)


BET Bromodomain Inhibitor

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Catalog No. A11783

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
GSK 1210151A 5mg A11783-5

Regular Price: €76.00

Special Price: €68.40

GSK 1210151A 10mg A11783-10

Regular Price: €114.00

Special Price: €102.60

GSK 1210151A 25mg A11783-25

Regular Price: €190.00

Special Price: €171.00

GSK 1210151A 50mg A11783-50

Regular Price: €342.00

Special Price: €307.80

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

GSK1210151A is a novel selective inhibitor of the bromodomain and extra terminal (BET) family proteins BRD2, BRD3, and BRD4.

GSK 1210151A (I-BET151)

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Publications citing Adooq Products
GSK 1210151A (I-BET151) Citations (1)
  • Momeny M, .et al. Inhibition of bromodomain and extraterminal domain reduces growth and invasive characteristics of chemoresistant ovarian carcinoma cells, Anticancer Drugs, 2018, Nov;29(10):1011-1020 PMID: 30096128

Chemical Information

Catalog Num A11783
Actions Inhibitor
M. Wt 415.4
Formula C23H21N5O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1300031-49-5
Synonyms GSK1210151A
SMILES CC1=C(C(=NO1)C)C2=C(C=C3C(=C2)N=CC4=C3N(C(=O)N4)[[email protected]](C)C5=CC=CC=N5)OC

Biological Activity

GSK1210151A is a novel selective inhibitor of the bromodomain and extra terminal (BET) family proteins BRD2, BRD3, and BRD4.
BRD3 (Cell-free assay) BRD2 (Cell-free assay) BRD4 (Cell-free assay)
0.25 μM0.5 μM0.79 μM


Solubility (25°C)* In vitro DMSO <1 mg/mL (<1 mM)
Water <1 mg/mL (<1 mM)
Ethanol 27 mg/mL (64.99 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.07 mL 120.37 mL 240.73mL
0.5 mM 4.81 mL 24.07 mL 48.15 mL
1 mM 2.41 mL 12.04 mL 24.07 mL
5 mM 0.48 mL 2.41 mL 4.81 mL

*The above data is based on the productmolecular weight 415.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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