GSK 1210151A (I-BET151)

Catalog No.: A11783

BET Bromodomain Inhibitor

GSK 1210151A (I-BET151)

GSK 1210151A (I-BET151) Chemical Structure

CAS NO. 1300031-49-5

GSK1210151A is a novel selective inhibitor of the bromodomain and extra terminal (BET) family proteins BRD2, BRD3, and BRD4.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $80.00

Special Price $72.00

10 mg

Regular Price: $120.00

Special Price $108.00

25 mg

Regular Price: $200.00

Special Price $180.00

50 mg

Regular Price: $360.00

Special Price $324.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

GSK1210151A is a novel selective inhibitor of the bromodomain and extra terminal (BET) family proteins BRD2, BRD3, and BRD4.
Targets
BRD3 (Cell-free assay) BRD2 (Cell-free assay) BRD4 (Cell-free assay)
0.25 μM0.5 μM0.79 μM
In vitro DMSO <1 mg/mL (<1 mM)
Water <1 mg/mL (<1 mM)
Ethanol 27 mg/mL (64.99 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.07 mL 120.37 mL 240.73 mL
0.5 mM 4.81 mL 24.07 mL 48.15 mL
1 mM 2.41 mL 12.04 mL 24.07 mL
5 mM 0.48 mL 2.41 mL 4.81 mL

*The above data is based on the productmolecular weight 415.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A11783
Actions Inhibitor
M. Wt 415.4
Formula C23H21N5O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1300031-49-5
Synonyms GSK1210151A
SMILES CC1=C(C(=NO1)C)C2=C(C=C3C(=C2)N=CC4=C3N(C(=O)N4)[[email protected]](C)C5=CC=CC=N5)OC

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