GSK-3326595 (EPZ015938)

Catalog No.: A16862

PRMT5 inhibitor

GSK-3326595 (EPZ015938)

GSK-3326595 (EPZ015938) Chemical Structure

CAS NO. 1616392-22-3

GSK3326595 is a potent, selective, reversible inhibitor of protein arginine methyltransferase 5 (PRMT5) with an IC50 of 6.2 nM.

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Package Price Qty
5 mg
$45.00
10 mg
$65.00
50 mg
$225.00
100 mg
$405.00
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Biological Activity

GSK3326595 is a potent, selective, reversible inhibitor of protein arginine methyltransferase 5 (PRMT5) with an IC50 of 6.2 nM.
In vitro DMSO 82 mg/mL (181.19 mM)
Water Insoluble
Ethanol 82 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.1 mL 110.49 mL 220.97 mL
0.5 mM 4.42 mL 22.1 mL 44.19 mL
1 mM 2.21 mL 11.05 mL 22.1 mL
5 mM 0.44 mL 2.21 mL 4.42 mL

*The above data is based on the productmolecular weight 452.55. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16862
Actions Inhibitor
CAS No. 1616392-22-3
Formula C24H32N6O3
M. Wt 452.55
Solubility DMSO
Purity >98%
Synonyms GSK3326595, GSK 3326595, EPZ-015938, EPZ 015938
SMILES O=C(C)N1CCC(NC2=NC=NC(C(NC[[email protected]](O)CN3CCC(C=CC=C4)=C4C3)=O)=C2)CC1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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