Biological Activity
GSK 525768A is the enantiomer compound of GSK 525762A, which is a potent small molecule inhibitor that disrupt the function of the BET family of bromodomains (Brd2, Brd3, and Brd4); GSK 525768A has NO activity towards BET.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 23.59 mL | 117.95 mL | 235.9 mL |
0.5 mM | 4.72 mL | 23.59 mL | 47.18 mL |
1 mM | 2.36 mL | 11.8 mL | 23.59 mL |
5 mM | 0.47 mL | 2.36 mL | 4.72 mL |
*The above data is based on the productmolecular weight 423.9. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A14134 |
---|---|
Actions | Inhibitor |
M. Wt | 423.9 |
Formula | C22H22ClN5O2 |
Solubility | DMSO |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 1260530-25-3 |
Synonyms | GSK525768A, GSK-525768A |
SMILES | CCNC(=O)C[[email protected]@H]1C2=NN=C(N2C3=C(C=C(C=C3)OC)C(=N1)C4=CC=C(C=C4)Cl)C |
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