GSK 525768A

Catalog No.: A14134

GSK 525768A

GSK 525768A Chemical Structure

CAS NO. 1260530-25-3

GSK 525768A is the enantiomer compound of GSK 525762A, which is a potent small molecule inhibitor that disrupt the function of the BET family of bromodomains (Brd2, Brd3, and Brd4); GSK 525768A has NO activity towards BET.

Availability: In stock

Package Price Qty
5 mg
$320.00
10 mg
$550.00
25 mg
$1,000.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

GSK 525768A is the enantiomer compound of GSK 525762A, which is a potent small molecule inhibitor that disrupt the function of the BET family of bromodomains (Brd2, Brd3, and Brd4); GSK 525768A has NO activity towards BET.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.59 mL 117.95 mL 235.9 mL
0.5 mM 4.72 mL 23.59 mL 47.18 mL
1 mM 2.36 mL 11.8 mL 23.59 mL
5 mM 0.47 mL 2.36 mL 4.72 mL

*The above data is based on the productmolecular weight 423.9. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A14134
Actions Inhibitor
M. Wt 423.9
Formula C22H22ClN5O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1260530-25-3
Synonyms GSK525768A, GSK-525768A
SMILES CCNC(=O)C[[email protected]@H]1C2=NN=C(N2C3=C(C=C(C=C3)OC)C(=N1)C4=CC=C(C=C4)Cl)C

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