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GSK 5959

BRPF1 bromodomain inhibitor

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Catalog No. A16092

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
GSK 5959 5mg A16092-5
€85.50
GSK 5959 10mg A16092-10
€142.50
GSK 5959 50mg A16092-50
€427.50

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

GSK 5959 is a potent, selective and cell permeable BRPF1 bromodomain inhibitor with IC50 ~ 80 nM. Exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains.

GSK 5959

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Chemical Information

Catalog Num A16092
Actions Inhibitor
M. Wt 394.48
Formula C22H26N4O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 901245-65-6
Synonyms GSK-5959, GSK5959
SMILES O=C(NC1=C(N2CCCCC2)C=C(N3C)C(N(C)C3=O)=C1)C4=CC=CC=C4OC

Biological Activity

Description
GSK 5959 is a potent, selective and cell permeable BRPF1 bromodomain inhibitor with IC50 ~ 80 nM. Exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.35 mL 126.75 mL 253.5mL
0.5 mM 5.07 mL 25.35 mL 50.7 mL
1 mM 2.53 mL 12.67 mL 25.35 mL
5 mM 0.51 mL 2.53 mL 5.07 mL

*The above data is based on the productmolecular weight 394.48. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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