GSK163090

Catalog No.: A15838

5-HT1A/B/D receptor antagonist

GSK163090

GSK163090 Chemical Structure

CAS NO. 844903-58-8

GSK163090 is a potent, selective, and orally active 5-HT1A/B/D receptor antagonist with pKi of 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3, respectively.

Availability: In stock

Package Price Qty
5 mg
$220.00
10 mg
$400.00
25 mg
$800.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

GSK163090 is a potent, selective, and orally active 5-HT1A/B/D receptor antagonist with pKi of 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.07 mL 120.33 mL 240.66 mL
0.5 mM 4.81 mL 24.07 mL 48.13 mL
1 mM 2.41 mL 12.03 mL 24.07 mL
5 mM 0.48 mL 2.41 mL 4.81 mL

*The above data is based on the productmolecular weight 415.53. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A15838
Actions Antagonist
M. Wt 415.53
Formula C25H29N5O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 844903-58-8
Synonyms GSK-163090, GSK 163090
SMILES CC1=NC2=C(C=C1)C(=CC=C2)N3CCN(CC3)CCC4=CC(=CC=C4)N5CCNC5=O

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