GSK163090

Catalog No.: A15838

5-HT1A/B/D receptor antagonist

GSK163090

GSK163090 Chemical Structure

CAS NO. 844903-58-8

GSK163090 is a potent, selective, and orally active 5-HT1A/B/D receptor antagonist with pKi of 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3, respectively.

Availability: In stock

Package Price Qty
5 mg
$220.00
10 mg
$400.00
25 mg
$800.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

GSK163090 is a potent, selective, and orally active 5-HT1A/B/D receptor antagonist with pKi of 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.07 mL 120.33 mL 240.66 mL
0.5 mM 4.81 mL 24.07 mL 48.13 mL
1 mM 2.41 mL 12.03 mL 24.07 mL
5 mM 0.48 mL 2.41 mL 4.81 mL

*The above data is based on the productmolecular weight 415.53. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15838
Actions Antagonist
CAS No. 844903-58-8
Formula C25H29N5O
M. Wt 415.53
Solubility DMSO
Purity >98%
Synonyms GSK-163090, GSK 163090
SMILES CC1=NC2=C(C=C1)C(=CC=C2)N3CCN(CC3)CCC4=CC(=CC=C4)N5CCNC5=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy GSK163090 | GSK163090 Supplier | purchase | cost | manufacturer | order | distributor | buy 844903-58-8| 844903-58-8 Supplier | purchase 844903-58-8 | 844903-58-8 cost | 844903-58-8 manufacturer | order 844903-58-8 | 844903-58-8 distributor
Rewards