Catalog No.: A12792
PERK inhibitor
GSK2606414 is an orally available, potent, and selective PERK inhibitor with IC50 of 0.4 nM.
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GSK2606414 5mg
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GSK2606414 10mg
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GSK2606414 25mg
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GSK2606414 50mg
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GSK2606414 10mM * 1mL in DMSO
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Adooq Products cited in reputable paper
Adooq's GSK2606414 has been cited by 2 publications
  • Linhao Xu, .et al. , Neural Plasticity, 2021, 23 Aug
  • Takashi Shimizu, .et al. , Sci Signal, 2021, Jan 26;14(667):eabb3616 PMID: 33500333
  • Biological Activity
    Discription GSK2606414 is an orally available, potent, and selective PERK inhibitor with IC50 of 0.4 nM.
    Target Value
    Product Information
    Catalog Num A12792
    Formula C24H20F3N5O
    Molecular Weight 451.44
    CAS Number 1337531-36-8
    SMILES CN1C=C(C2=C1N=CN=C2N)C3=CC4=C(C=C3)N(CC4)C(=O)CC5=CC(=CC=C5)C(F)(F)F
    Synonyms GSK-2606414, GSK 2606414

    Store lyophilized at -20ºC, keep desiccated.
    In lyophilized form, the chemical is stable for 36 months.
    In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

    In vitro (25°C) DMSO 87 mg/mL (192.71 mM)
    Water Insoluble
    Ethanol 18 mg/mL (39.87 mM)
    In vivo 5% DMSO+45% PEG 300+ddH2O 19 mg/mL
    * <1 mg/ml means slightly soluble or insoluble.
    * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
    Preparing Stock Solutions
    Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
    0.1 mM 22.15 mL 110.76 mL 221.51 mL
    0.5 mM 4.43 mL 22.15 mL 44.3 mL
    1 mM 2.22 mL 11.08 mL 22.15 mL
    5 mM 0.44 mL 2.22 mL 4.43 mL
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    Calculate the dilution required to prepare a stock solution.
    This equation is commonly abbreviated as: C1V1 = C2V2

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