Biological Activity
GSK2973980A is a potent and selective Acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitor with an IC50 of 3 nM.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 18.71 mL | 93.56 mL | 187.12 mL |
0.5 mM | 3.74 mL | 18.71 mL | 37.42 mL |
1 mM | 1.87 mL | 9.36 mL | 18.71 mL |
5 mM | 0.37 mL | 1.87 mL | 3.74 mL |
*The above data is based on the productmolecular weight 534.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A20060 |
---|---|
Actions | Inhibitor |
CAS No. | 2219321-25-0 |
Formula | C25H19F5N4O4 |
M. Wt | 534.43 |
Purity | >98% |
Synonyms | GSK 2973980A, GSK-2973980A |
SMILES | FC1=C(F)C=C(NC(NC2=CN=C(C3=CC(CC[[email protected]](CC(O)=O)(CC(F)(F)F)C4=O)=C4C=C3)C=N2)=O)C=C1 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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