GSK2973980A

Catalog No.: A20060

DGAT1 inhibitor

GSK2973980A

GSK2973980A Chemical Structure

CAS NO. 2219321-25-0

GSK2973980A is a potent and selective Acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitor with an IC50 of 3 nM.

Availability: In stock

Package Price Qty
5 mg
$350.00
10 mg
$650.00
50 mg
$2,000.00
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Biological Activity

GSK2973980A is a potent and selective Acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitor with an IC50 of 3 nM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.71 mL 93.56 mL 187.12 mL
0.5 mM 3.74 mL 18.71 mL 37.42 mL
1 mM 1.87 mL 9.36 mL 18.71 mL
5 mM 0.37 mL 1.87 mL 3.74 mL

*The above data is based on the productmolecular weight 534.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A20060
Actions Inhibitor
CAS No. 2219321-25-0
Formula C25H19F5N4O4
M. Wt 534.43
Solubility DMSO
Purity >98%
Synonyms GSK 2973980A, GSK-2973980A
SMILES FC1=C(F)C=C(NC(NC2=CN=C(C3=CC(CC[[email protected]](CC(O)=O)(CC(F)(F)F)C4=O)=C4C=C3)C=N2)=O)C=C1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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