GW 9662

Catalog No.: A11984

PPARγ antagonist

GW 9662

GW 9662 Chemical Structure

CAS NO. 22978-25-2

GW 9662 is a selective PPARγ antagonist (IC50 values are 3.3, 32 and 2000 nM for PPARγ, PPARα and PPARδ respectively).

Availability: In stock

Package Price Qty
10 mg

Regular Price: $60.00

Special Price $54.00

25 mg

Regular Price: $90.00

Special Price $81.00

50 mg

Regular Price: $120.00

Special Price $108.00

100 mg

Regular Price: $220.00

Special Price $198.00

10mM * 1mL in DMSO

Regular Price: $50.00

Special Price $45.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

GW 9662 is a selective PPARγ antagonist (IC50 values are 3.3, 32 and 2000 nM for PPARγ, PPARα and PPARδ respectively).
Targets
PPARγ (Cell-free assay) PPARα (Cell-free assay) PPARδ (Cell-free assay)
3.3 nM32 nM2 μM
In vitro (25°C) DMSO 55 mg/mL (198.78 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 1% DMSO/30% polyethylene glycol/1% Tween 80 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 36.14 mL 180.71 mL 361.43 mL
0.5 mM 7.23 mL 36.14 mL 72.29 mL
1 mM 3.61 mL 18.07 mL 36.14 mL
5 mM 0.72 mL 3.61 mL 7.23 mL

*The above data is based on the productmolecular weight 276.68. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A11984
Actions Antagonist
M. Wt 276.68
Formula C13H9N2O3Cl
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 22978-25-2
Synonyms GW9662, GW-9662
SMILES C1=CC=C(C=C1)NC(=O)C2=C(C=CC(=C2)[N+](=O)[O-])Cl

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