GW 9662

Catalog No.: A11984

PPARγ antagonist

GW 9662

GW 9662 Chemical Structure

CAS NO. 22978-25-2

GW 9662 is a selective PPARγ antagonist (IC50 values are 3.3, 32 and 2000 nM for PPARγ, PPARα and PPARδ respectively).

Availability: In stock

Package Price Qty
10 mg
$60.00
25 mg
$90.00
50 mg
$120.00
100 mg
$220.00
10mM * 1mL in DMSO
$50.00
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Biological Activity

GW 9662 is a selective PPARγ antagonist (IC50 values are 3.3, 32 and 2000 nM for PPARγ, PPARα and PPARδ respectively).
Targets
PPARγ (Cell-free assay) PPARα (Cell-free assay) PPARδ (Cell-free assay)
3.3 nM32 nM2 μM
In vitro (25°C) DMSO 48 mg/mL (173.48 mM)
Water Insoluble
Ethanol Insoluble
In vivo 5% DMSO+corn oil 8 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 36.14 mL 180.71 mL 361.43 mL
0.5 mM 7.23 mL 36.14 mL 72.29 mL
1 mM 3.61 mL 18.07 mL 36.14 mL
5 mM 0.72 mL 3.61 mL 7.23 mL

*The above data is based on the productmolecular weight 276.68. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11984
Actions Antagonist
CAS No. 22978-25-2
Formula C13H9N2O3Cl
M. Wt 276.68
Purity >98%
Synonyms GW9662, GW-9662
SMILES C1=CC=C(C=C1)NC(=O)C2=C(C=CC(=C2)[N+](=O)[O-])Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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