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Biological Activity
GW842166X is a selective non-cannabinoid CB2 receptor agonist, which is undergoing clinical development as a novel oral treatment for inflammatory pain
Targets
| CB2 | ||||
| 63 nM(EC50) |
| In vitro (25°C) | DMSO | 18 mg/mL (40.06 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
| In vivo | 30% propylene glycol, 5% Tween 80, 65% D5W | 28 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 22.26 mL | 111.3 mL | 222.59 mL |
| 0.5 mM | 4.45 mL | 22.26 mL | 44.52 mL |
| 1 mM | 2.23 mL | 11.13 mL | 22.26 mL |
| 5 mM | 0.45 mL | 2.23 mL | 4.45 mL |
*The above data is based on the productmolecular weight 449.25. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A11253 |
|---|---|
| Actions | Agonist |
| CAS No. | 666260-75-9, 956013-38-0 |
| Formula | C18H17Cl2F3N4O2 |
| M. Wt | 449.25 |
| Purity | >98% |
| SMILES | C1COCCC1CNC(=O)C2=CN=C(N=C2C(F)(F)F)NC3=C(C=C(C=C3)Cl)Cl |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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Contact information
United StatesAdooq Bioscience
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Email: [email protected]
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