GW842166X

Catalog No.: A11253

CB2 receptor agonist

GW842166X Chemical Structure

CAS NO. 666260-75-9, 956013-38-0

GW842166X is a selective non-cannabinoid CB2 receptor agonist, which is undergoing clinical development as a novel oral treatment for inflammatory pain

Availability: In stock

Package Price Qty
5 mg
$60.00
10 mg
$100.00
25 mg
$200.00
10mM * 1mL in DMSO
$113.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

GW842166X is a selective non-cannabinoid CB2 receptor agonist, which is undergoing clinical development as a novel oral treatment for inflammatory pain
Targets
CB2
63 nM(EC50)
In vitro (25°C) DMSO 20 mg/mL (44.51 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.26 mL 111.3 mL 222.59 mL
0.5 mM 4.45 mL 22.26 mL 44.52 mL
1 mM 2.23 mL 11.13 mL 22.26 mL
5 mM 0.45 mL 2.23 mL 4.45 mL

*The above data is based on the productmolecular weight 449.25. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11253
Actions Agonist
M. Wt 449.25
Formula C18H17Cl2F3N4O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 666260-75-9, 956013-38-0
Synonyms N/A
SMILES C1COCCC1CNC(=O)C2=CN=C(N=C2C(F)(F)F)NC3=C(C=C(C=C3)Cl)Cl

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy GW842166X | GW842166X Supplier | purchase GW842166X | GW842166X cost | GW842166X manufacturer | order GW842166X | GW842166X distributor | buy 666260-75-9, 956013-38-0| 666260-75-9, 956013-38-0 Supplier | purchase 666260-75-9, 956013-38-0 | 666260-75-9, 956013-38-0 cost | 666260-75-9, 956013-38-0 manufacturer | order 666260-75-9, 956013-38-0 | 666260-75-9, 956013-38-0 distributor
Rewards