GW843682X

Catalog No.: A11438

PLK1/PLK3 inhibitor

GW843682X

GW843682X Chemical Structure

CAS NO. 660868-91-7

GW843682X is a selective inhibitor of polo-like kinase 1 (PLK1) and polo-like kinase 3 (PLK3) (IC50 values are 2.2 and 9.1 nM respectively).

Availability: In stock

Package Price Qty
5 mg
$70.00
10 mg
$120.00
25 mg
$250.00
50 mg
$450.00
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.
  • Kanada F, .et al. Histone acetyltransferase and Polo-like kinase 3 inhibitors prevent rat galactose-induced cataract, Sci Rep, 2019, Dec 27;9(1):20085 PMID: 31882756

Biological Activity

GW843682X is a selective inhibitor of polo-like kinase 1 (PLK1) and polo-like kinase 3 (PLK3) (IC50 values are 2.2 and 9.1 nM respectively).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.94 mL 104.72 mL 209.44 mL
0.5 mM 4.19 mL 20.94 mL 41.89 mL
1 mM 2.09 mL 10.47 mL 20.94 mL
5 mM 0.42 mL 2.09 mL 4.19 mL

*The above data is based on the productmolecular weight 477.46. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11438
Actions Inhibitor
CAS No. 660868-91-7
Formula C22H18F3N3O4S
M. Wt 477.46
Purity >98%
SMILES COC1=C(C=C2C(=C1)N=CN2C3=CC(=C(S3)C(=O)N)OCC4=CC=CC=C4C(F)(F)F)OC
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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